Protective effect of methanol extract of Uncaria rhynchophylla against excitotoxicity induced by N-methyl-D-aspartate in rat hippocampus.

نویسندگان

  • Jongseok Lee
  • Dongwook Son
  • Pyeongjae Lee
  • Dae-Keun Kim
  • Min-Chul Shin
  • Mi-Hyeon Jang
  • Chang-Ju Kim
  • Yong-Sik Kim
  • Sun-Yeou Kim
  • Hocheol Kim
چکیده

Uncaria rhynchophylla is a medicinal herb used for convulsive disorders in Oriental medicine. In this study, the effect of the methanol extract of Uncaria rhynchophylla against N-methyl-D-aspartate (NMDA)-induced excitotoxicity was investigated. Pretreatment with the extract of Uncaria rhynchopylla reduced the degree of neuronal damage induced by NMDA exposure in cultured hippocampal slices. In the patch clamp study, Uncaria rhynchophylla significantly inhibited NMDA receptor-activated ion current in acutely dissociated hippocampal CA1 neurons. These results indicate that Uncaria rhynchophylla offers protection against NMDA-induced neuronal injury and inhibitory action on NMDA receptor-mediated ion current may be a mechanism behind the neuroprotective effect of Uncaria rhynchophylla.

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عنوان ژورنال:
  • Journal of pharmacological sciences

دوره 92 1  شماره 

صفحات  -

تاریخ انتشار 2003